SCHEMBL12933697

SCHEMBL12933697

CC(C)CNC(C)c1nc2cc(Cl)ccc2c(=O)n1Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 6/20 0.50
CYP3A4 P08684 2/20 0.50
MAP1LC3B Q9GZQ8 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
CYP2C19 P33261 1/20 0.50
KCNH2 Q12809 1/20 0.50
ALOX5AP P20292 1/20 0.46
EGFR P00533 1/20 0.45
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
PDE1C Q14123 1/20 0.43
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPK8 P45983 1/20 0.42
MAPK9 P45984 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12963732 0.90 TDP1 (0.51) KIF11CYP3A4MAP1LC3BTDP1CYP2C19
SCHEMBL12933365 0.89 KIF11 (0.49) KIF11CYP3A4MAP1LC3BTDP1CYP2C19
SCHEMBL16645078 0.83 KIF11 (0.56) KIF11CYP3A4MAP1LC3BTDP1CYP2C19
SCHEMBL4283747 0.81 KIF11 (0.56) KIF11CYP3A4MAP1LC3BTDP1CYP2C19
SCHEMBL5648396 0.81 KIF11 (0.56) KIF11CYP3A4MAP1LC3BTDP1CYP2C19
SCHEMBL4517998 0.81 KIF11 (0.54) KIF11CYP3A4MAP1LC3BTDP1CYP2C19
SCHEMBL4519529 0.81 KIF11 (0.56) KIF11CYP3A4MAP1LC3BTDP1CYP2C19
SCHEMBL12963255 0.81 KIF11 (0.51) KIF11CYP3A4MAP1LC3BTDP1CYP2C19
SCHEMBL4522589 0.80 KIF11 (0.48) KIF11CYP3A4MAP1LC3BTDP1CYP2C19
SCHEMBL4620734 0.80 KIF11 (0.57) KIF11CYP3A4MAP1LC3BTDP1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7868204-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2011-01-11 US disclosed
US-7838520-B2 Inhibitors of histone deacetylase METHYLGENE, INC. (CA) 2010-11-23 US disclosed
US-7595343-B2 Inhibitors of histone deacetylase METHYLGENE, INC. (CA) 2009-09-29 US disclosed