SCHEMBL12969725

SCHEMBL12969725

Nc1ncnc2c1sc1nc(-c3cc4ccccc4o3)cc(-c3ccccc3)c12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIMK1 P53667 7/20 0.51
CDC7 O00311 7/20 0.45
DBF4 Q9UBU7 6/20 0.45
CLK1 P49759 2/20 0.45
GRM4 Q14833 1/20 0.44
MAPT P10636 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
PLK4 O00444 2/20 0.42
AURKA O14965 2/20 0.42
ROCK2 O75116 2/20 0.42
PIM1 P11309 2/20 0.42
PRKACA P17612 2/20 0.42
RPS6KB1 P23443 2/20 0.42
CDK2 P24941 2/20 0.42
MARK3 P27448 2/20 0.42
FLT4 P35916 2/20 0.42
KDR P35968 2/20 0.42
CSNK1D P48730 2/20 0.42
GSK3A P49840 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4899938 0.84 LIMK1 (0.66) LIMK1CDC7DBF4CLK1MAPT
SCHEMBL12969721 0.81 LIMK1 (0.65) LIMK1CDC7DBF4CLK1GRM4
SCHEMBL4900157 0.78 HPGD (0.62) LIMK1CDC7DBF4CLK1MAPT
SCHEMBL4899880 0.78 KDM4E (0.62) LIMK1CDC7DBF4CLK1MAPT
SCHEMBL4905558 0.78 CDC7 (0.66) LIMK1CDC7DBF4CLK1MAPT
SCHEMBL4894356 0.78 HPGD (0.58) LIMK1CLK1MAPT
SCHEMBL4899003 0.77 MEN1 (0.59) LIMK1CDC7DBF4CLK1MAPT
SCHEMBL4902783 0.76 PPARG (0.64) LIMK1CDC7DBF4CLK1PLK4
SCHEMBL259291 0.73 CDC7 (0.66) LIMK1CDC7DBF4CLK1MAPT
SCHEMBL4899997 0.71 MAPT (0.50) LIMK1MAPTMKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012131297-A1 PYRIDO [3',2' :4,5] THIENO [3, 2-D] PYRIMIDIN- 4 - YLAMINE DERIVATIVES AND THEIR THERAPEUTICAL USE BAELL JONATHAN BAYLDON (AU) 2012-10-04 WO disclosed