SCHEMBL12987693

SCHEMBL12987693

CCc1nc2nc3ccccc3c(=O)n2c2c1CCC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.39
KDM4E B2RXH2 6/20 0.39
HSD17B10 Q99714 3/20 0.39
HPGD P15428 3/20 0.39
LMNA P02545 2/20 0.39
USP2 O75604 1/20 0.39
CYP1A2 P05177 1/20 0.39
BCHE P06276 1/20 0.39
CFTR P13569 1/20 0.39
ALOX15 P16050 1/20 0.39
ACHE P22303 1/20 0.39
HKDC1 Q2TB90 1/20 0.39
GOPC Q9HD26 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 4/20 0.39
PDE5A O76074 2/20 0.39
MAPT P10636 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12987717 0.98 KDM4E (0.41) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL12987105 0.85 PDE5A (0.39) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL12987735 0.81 KDM4E (0.40) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL12987270 0.78 MEN1 (0.40) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL12987397 0.77 KDM4E (0.51) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL12987706 0.72 PDE4A (0.44) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL12987385 0.70 TNKS2 (0.40) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL12987559 0.68 ALDH1A1 (0.38) ALDH1A1KDM4EHSD17B10HPGDLMNA
SCHEMBL12987529 0.67 ATM (0.35) ALDH1A1HPGDBCHEACHESMN1; SMN2
SCHEMBL10287048 0.63 CYP1A2 (0.46) ALDH1A1KDM4EHSD17B10HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7855214-B2 Fused cyclic systems useful as inhibitors of TEC family protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-12-21 US disclosed