SCHEMBL12995249

SCHEMBL12995249

Cc1oc(C(=O)O)cc1Br

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 3/20 0.52
CHRNA4 P43681 2/20 0.51
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MCL1 Q07820 1/20 0.44
PIM1 P11309 2/20 0.43
PTGER4 P35408 4/20 0.42
DAO P14920 1/20 0.42
HCAR2 Q8TDS4 1/20 0.41
MAPT P10636 2/20 0.41
ALDH1A1 P00352 2/20 0.41
POLB P06746 2/20 0.41
HSD17B10 Q99714 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MEN1 O00255 1/20 0.41
ALOX15 P16050 1/20 0.41
LIG1 P18858 1/20 0.41
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1198612 0.78 MAPT (0.53) CHRNA4KMT2AKDM4EMAPTALDH1A1
SCHEMBL700764 0.77 APEX1 (0.55) APEX1KMT2AKDM4EPTGER4DAO
SCHEMBL274316 0.77 CHRNA4 (0.49) APEX1CHRNA4KMT2AKDM4EMCL1
SCHEMBL14620144 0.76 APEX1 (0.53) APEX1KMT2AKDM4EPTGER4DAO
SCHEMBL20582083 0.74 KMT2A (0.48) APEX1KMT2AKDM4EMCL1PIM1
SCHEMBL29952181 0.74 APEX1 (0.52) APEX1KMT2AKDM4EPIM1PTGER4
SCHEMBL28651161 0.74 DAO (0.63) APEX1KMT2AKDM4EMCL1PIM1
SCHEMBL27770730 0.74 POLB (0.56) APEX1KMT2AKDM4EMCL1PIM1
SCHEMBL9311435 0.72 KDM4E (0.52) APEX1KMT2AKDM4EPTGER4DAO
SCHEMBL22638673 0.72 APEX1 (0.46) APEX1KMT2AKDM4EMCL1PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2264017-A1 HETEROCYCLIC DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2010-12-22 EP disclosed