SCHEMBL13015490

SCHEMBL13015490

COc1c(C)ncc(C)c1C

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AGXT P21549 1/20 0.44
CCR1 P32246 1/20 0.38
CCR5 P51681 1/20 0.38
CCR8 P51685 1/20 0.38
HSP90AB1 P08238 2/20 0.35
MAOA P21397 1/20 0.34
HSP90AA1 P07900 1/20 0.34
TDP1 Q9NUW8 1/20 0.31
ACHE P22303 1/20 0.31
DHFR P00374 1/20 0.31
PDE10A Q9Y233 2/20 0.30
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16921630 0.83 AGXT (0.46) AGXTCCR1CCR5CCR8HSP90AB1
SCHEMBL94923 0.81 AGXT (0.53) AGXTCCR1CCR5CCR8HSP90AB1
SCHEMBL29039529 0.79 AGXT (0.52) AGXTCCR1CCR5CCR8HSP90AB1
SCHEMBL29736023 0.79 AGXT (0.52) AGXTCCR1CCR5CCR8HSP90AB1
Hydrochloric Acid SCHEMBL28303939 0.79 AGXT (0.52) AGXTCCR1CCR5CCR8HSP90AB1
SCHEMBL1731691 0.77 CCR1 (0.35) AGXTCCR1CCR5CCR8HSP90AB1
SCHEMBL12207313 0.77 AGXT (0.38) AGXTHSP90AB1MAOAHSP90AA1
SCHEMBL10440855 0.74 AGXT (0.51) AGXTCCR1CCR5CCR8HSP90AB1
SCHEMBL2740251 0.73 AGXT (0.42) AGXTMAOA
SCHEMBL192172 0.73 AGXT (0.42) AGXTHSP90AB1MAOAHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2266958-A1 Antiviral agent SHIONOGI & CO., LTD. (JP) 2010-12-29 EP disclosed
US-20070185064-A1 2-Aminopurine Analogs Having HSP90-Inhibiting Activity CONFORMA THERAPEUTICS CORPORATION (US) 2007-08-09 US disclosed
US-20070185064-A1 2-Aminopurine Analogs Having HSP90-Inhibiting Activity CONFORMA THERAPEUTICS CORPORATION (US) 2007-08-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070185064-A1 2-Aminopurine Analogs Having HSP90-Inhibiting Activity HSP90AB2P, HSP90AB1, HSP90AA1 AGXT 1906/4885CCR1 4568/4885CCR5 4618/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.