SCHEMBL13019683

SCHEMBL13019683

COc1ccccc1C(F)F

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.57
CA2 P00918 4/20 0.57
CA7 P43166 2/20 0.57
CA9 Q16790 2/20 0.57
CA12 O43570 1/20 0.57
CA4 P22748 1/20 0.57
CA14 Q9ULX7 1/20 0.57
IDO1 P14902 3/20 0.47
TDO2 P48775 1/20 0.47
ALDH1A1 P00352 3/20 0.46
TDP1 Q9NUW8 2/20 0.46
TP53 P04637 1/20 0.46
TSHR P16473 1/20 0.46
ADRA2B P18089 1/20 0.46
PTGS1 P23219 1/20 0.46
HTT P42858 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
MAPK1 P28482 1/20 0.44
ACHE P22303 1/20 0.44
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29005947 0.82 CA1 (0.48) CA1CA2CA7CA9CA12
SCHEMBL22827469 0.82 KRAS (0.44) CA1CA2CA7CA9CA12
SCHEMBL22827153 0.82 CA1 (0.42) CA1CA2CA7CA9CA12
SCHEMBL8879882 0.81 CA1 (0.52) CA1CA2CA7CA9CA12
SCHEMBL27772307 0.81 CA1 (0.52) CA1CA2CA7CA9CA12
SCHEMBL27772296 0.81 CA1 (0.52) CA1CA2CA7CA9CA12
SCHEMBL28238041 0.81 CA1 (0.52) CA1CA2CA7CA9CA12
SCHEMBL27999515 0.81 ALDH1A1 (0.43) CA1CA2CA7CA9CA12
SCHEMBL17593428 0.79 IRAK4 (0.44) CA1CA2CA7CA9ALDH1A1
SCHEMBL31511214 0.79 ALDH1A1 (0.52) ALDH1A1TDP1L3MBTL1MAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9475756-B2 Difluoromethylation of aryl and vinyl iodides THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-10-25 US disclosed
US-9475756-B2 Difluoromethylation of aryl and vinyl iodides THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-10-25 US disclosed
US-9475756-B2 Difluoromethylation of aryl and vinyl iodides THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-10-25 US disclosed
US-20150045580-A1 DIFLUOROMETHYLATION OF ARYL AND VINYL IODIDES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-02-12 US disclosed
US-20150045580-A1 DIFLUOROMETHYLATION OF ARYL AND VINYL IODIDES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-02-12 US disclosed
US-20150045580-A1 DIFLUOROMETHYLATION OF ARYL AND VINYL IODIDES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-02-12 US disclosed
WO-2013134296-A1 DIFLUOROMETHYLATION OF ARYL AND VINYL IODIDES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2013-09-12 WO disclosed
CN-101547922-B Pyrido[4,3-d]pyrimidin-4(3h)-one derivatives as calcium receptor antagonists PFIZER PROD INC 2012-06-20 CN disclosed
US-20100331310-A1 BICYCLOAMINE DERIVATIVES EISAI R&D MANAGEMENT CO., LTD. (JP) 2010-12-30 US disclosed
CN-101910169-A Bicyclic amine derivatives EISAI R&D MAN CO LTD 2010-12-08 CN disclosed
CN-101547922-A Pyrido[4,3-d]pyrimidin-4(3H)-one derivatives as calcium receptor antagonists PFIZER PRODUCT INC (US) 2009-09-30 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100331310-A1 BICYCLOAMINE DERIVATIVES SCN1B, KCNJ2, KCNH2 CA1 2021/4885CA2 883/4885CA7 3048/4885
US-20150045580-A1 DIFLUOROMETHYLATION OF ARYL AND VINYL IODIDES CUL2, CUL3, CYP4F2 CA1 3188/4885CA2 3435/4885CA7 3209/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.