SCHEMBL1302019

SCHEMBL1302019

Nc1ccc2c(c1N)C(=O)C(=O)c1ccccc1-2

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.78
MAOB P27338 1/20 0.78
ADORA2A P29274 5/20 0.59
CSNK1A1 P48729 2/20 0.59
CSNK1D P48730 2/20 0.59
CSNK1G1 Q9HCP0 2/20 0.59
FGR P09769 1/20 0.59
PIM1 P11309 1/20 0.59
DYRK1A Q13627 1/20 0.59
HIPK2 Q9H2X6 1/20 0.59
MEN1 O00255 8/20 0.54
KMT2A Q03164 8/20 0.54
POLB P06746 7/20 0.54
SMN1; SMN2 Q16637 6/20 0.54
MAPK1 P28482 6/20 0.54
PTPRC P08575 5/20 0.54
MAPT P10636 5/20 0.54
RAB9A P51151 5/20 0.54
LMNA P02545 4/20 0.54
NPC1 O15118 4/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3740221 0.96 MAOA (0.85) MAOAMAOBADORA2ACSNK1A1CSNK1D
SCHEMBL31177128 0.96 MAOA (0.85) MAOAMAOBADORA2ACSNK1A1CSNK1D
SCHEMBL30129869 0.88 MAOA (1.00) MAOAMAOBADORA2ACSNK1A1CSNK1D
SCHEMBL487001 0.88 MAOA (1.00) MAOAMAOBADORA2ACSNK1A1CSNK1D
Ammonia Solution, Strong SCHEMBL6046897 0.86 MAOA (0.96) MAOAMAOBADORA2ACSNK1A1CSNK1D
SCHEMBL29372739 0.82 MAOA (0.57) MAOAMAOBADORA2ACSNK1A1CSNK1D
SCHEMBL475599 0.82 MAOA (0.57) MAOAMAOBADORA2ACSNK1A1CSNK1D
SCHEMBL1447534 0.82 MAOA (0.57) MAOAMAOBADORA2ACSNK1A1CSNK1D
SCHEMBL28827042 0.81 MAOA (0.86) MAOAMAOBADORA2ACSNK1A1CSNK1D
Methoxymethane SCHEMBL11741879 0.81 MAOA (0.86) MAOAMAOBADORA2ACSNK1A1CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118359781-A Ferrocene group-containing polymer, preparation method and application thereof 南开大学 2024-07-19 CN disclosed
EP-2391925-B1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KK (JP) 2018-09-19 EP disclosed
US-8465889-B2 Electrophotographic photosensitive member, process cartridge, and electrophotographic apparatus CANON KABUSHIKI KAISHA (JP) 2013-06-18 US disclosed
US-8435706-B2 2013-05-07 US disclosed
EP-2391925-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS Canon Kabushiki Kaisha (JP) 2011-12-07 EP disclosed
US-20110268472-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2011-11-03 US disclosed
WO-2010087520-A1 ELECTROPHOTOGRAPHIC PHOTOSENSITIVE MEMBER, PROCESS CARTRIDGE, AND ELECTROPHOTOGRAPHIC APPARATUS CANON KABUSHIKI KAISHA (JP) 2010-08-05 WO disclosed
US-4186263-A MOLDABLE AT LOWER TEMPERATURES THAN IN PRIOR ART STANDARD OIL COMPANY (INDIANA) (US) 1980-01-29 US disclosed