SCHEMBL13030722

SCHEMBL13030722

Cc1ncc(-c2ccc(Oc3ccc(F)cc3)cc2)[nH]1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN4A P35499 2/20 0.51
LTA4H P09960 1/20 0.48
CYP2A6 P11509 1/20 0.45
SCN2A Q99250 2/20 0.41
SCN10A Q9Y5Y9 4/20 0.40
KCNH2 Q12809 3/20 0.40
SCN1A P35498 1/20 0.40
SCN5A Q14524 1/20 0.40
SCN9A Q15858 1/20 0.40
SCN8A Q9UQD0 1/20 0.40
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
GFER P55789 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
BACE1 P56817 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7483325 0.90 CYP2A6 (0.53) CYP2A6ALDH1A1MAPTHPGDGFER
SCHEMBL13159520 0.80 CYP2A6 (0.49) SCN4ALTA4HCYP2A6SCN2ASCN10A
SCHEMBL17269665 0.80 SCN2A (0.61) SCN4ACYP2A6SCN2ASCN10AMAPT
SCHEMBL15747113 0.75 CYP2A6 (0.56) CYP2A6SCN2AALDH1A1MAPTHPGD
SCHEMBL17066735 0.73 CYP2A6 (0.55) CYP2A6SCN2AALDH1A1MAPTGFER
SCHEMBL17066723 0.73 CYP2A6 (0.55) CYP2A6SCN2AALDH1A1MAPTGFER
SCHEMBL13115506 0.73 SCN2A (0.75) SCN2ASCN10A
SCHEMBL24427567 0.72 CYP2A6 (0.53) LTA4HCYP2A6SCN2ASCN10AALDH1A1
SCHEMBL7904690 0.72 POLB (0.61) LTA4HCYP2A6SCN2ASCN10ASCN5A
SCHEMBL28559389 0.72 CYP2A6 (0.53) CYP2A6SCN2ASCN10AGFERPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2266960-B1 Aryl-substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles as anticonvulsants EURO CELTIQUE SA (LU) 2014-01-22 EP disclosed
EP-2266960-A2 Aryl-substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles as anticonvulsants EURO-CELTIQUE S.A. (LU) 2010-12-29 EP disclosed
EP-1173169-B1 ARYL SUBSTITUTED PYRAZOLES, IMIDAZOLES, OXAZOLES, THIAZOLES AND PYRROLES, AND THE USE THEREOF EURO CELTIQUE SA (LU) 2010-05-12 EP disclosed