SCHEMBL13045239

SCHEMBL13045239

C[C@H]1CN(C[C@H](Cc2ccccc2)C(=O)O)CCC1(C)c1cccc(C(N)=O)c1

nearest known ligand 0.78

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 17/20 0.78
OPRD1 P41143 12/20 0.78
OPRK1 P41145 13/20 0.74
KCNE1 P15382 1/20 0.62
KCNQ1 P51787 1/20 0.62
CACNA1C Q13936 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3763241 1.00 OPRM1 (0.78) OPRM1OPRD1OPRK1KCNE1KCNQ1
SCHEMBL1705349 1.00 OPRM1 (0.78) OPRM1OPRD1OPRK1KCNE1KCNQ1
SCHEMBL12997002 1.00 OPRM1 (0.78) OPRM1OPRD1OPRK1KCNE1KCNQ1
SCHEMBL1705344 1.00 OPRM1 (0.78) OPRM1OPRD1OPRK1KCNE1KCNQ1
SCHEMBL3726859 0.94 OPRM1 (0.74) OPRM1OPRD1OPRK1KCNE1KCNQ1
SCHEMBL12587737 0.94 OPRM1 (0.73) OPRM1OPRD1OPRK1KCNE1KCNQ1
SCHEMBL12997060 0.94 OPRM1 (0.73) OPRM1OPRD1OPRK1KCNE1KCNQ1
SCHEMBL12555224 0.94 OPRM1 (0.73) OPRM1OPRD1OPRK1KCNE1KCNQ1
SCHEMBL1217627 0.93 OPRM1 (0.81) OPRM1OPRD1OPRK1KCNE1KCNQ1
SCHEMBL1705321 0.92 OPRM1 (0.70) OPRM1OPRD1OPRK1KCNE1KCNQ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010144446-A1 (S) -2-BENZYL-3- ( (3R, 4R) -4- (3 -CARBAMO YLPHENYL) -3, 4-DIMETHYLPIPERIDINYL) PROPANOIC ACID AND SALT THEROF AS ANTAGONISTS OF THE OPIOID RECEPTORS ADOLOR CORPORATION (US) 2010-12-16 WO disclosed