SCHEMBL13048632

SCHEMBL13048632

CNC(=O)CCc1cccc(Nc2nc(NC3CC3)c3c(S(C)(=O)=O)n[nH]c3n2)c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 7/20 0.43
IRAK4 Q9NWZ3 1/20 0.39
PKMYT1 Q99640 1/20 0.39
PIK3CD O00329 1/20 0.38
PIK3CA P42336 1/20 0.38
PIK3CB P42338 1/20 0.38
PIK3CG P48736 1/20 0.38
SYK P43405 3/20 0.37
EML4 Q9HC35 1/20 0.36
ALK Q9UM73 1/20 0.36
PDE5A O76074 1/20 0.36
NEK2 P51955 2/20 0.36
CSNK2A1 P68400 1/20 0.36
JAK2 O60674 2/20 0.36
JAK1 P23458 2/20 0.36
JAK3 P52333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13048635 0.92 NEK2 (0.44) IGF1RIRAK4PKMYT1PIK3CDPIK3CA
SCHEMBL13048831 0.86 SYK (0.42) SYKJAK2
SCHEMBL13048603 0.86 SYK (0.48) SYKJAK2
SCHEMBL13048648 0.82 PIK3CD (0.43) PIK3CDPIK3CAPIK3CBPIK3CGSYK
SCHEMBL13048641 0.81 SYK (0.45) PIK3CDPIK3CAPIK3CBPIK3CGSYK
SCHEMBL13048627 0.81 PIK3CD (0.41) IRAK4PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL13048827 0.80 SYK (0.43) IGF1RIRAK4SYKEML4ALK
SCHEMBL13048643 0.79 FLT3 (0.41) IGF1RPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL13048825 0.78 PIK3CG (0.45) PIK3CDPIK3CAPIK3CBPIK3CGSYK
SCHEMBL13048565 0.78 SYK (0.56) SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100298557-A1 PYRAZOLOPYRIMIDINE COMPOUND TAISHO PHARMACEUTICAL CO., LTD (JP) 2010-11-25 US disclosed
US-20100298557-A1 PYRAZOLOPYRIMIDINE COMPOUND TAISHO PHARMACEUTICAL CO., LTD (JP) 2010-11-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100298557-A1 PYRAZOLOPYRIMIDINE COMPOUND SYK, LCK, FYN IGF1R 1118/4885IRAK4 117/4885PKMYT1 300/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.