SCHEMBL13055052

SCHEMBL13055052

CN1CCN(C(=O)OCc2ccccc2)CC1c1cc(Nc2n[nH]c3ccccc23)nc(-c2ccc3[nH][nH]c(=O)c3c2C(F)(F)F)n1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 1/20 0.38
USP30 Q70CQ3 1/20 0.36
MAPK10 P53779 13/20 0.35
MAPK8 P45983 7/20 0.35
MAPK1 P28482 1/20 0.34
PARP1 P09874 2/20 0.33
TNKS O95271 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
PARP2 Q9UGN5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL802156 0.87 FLT3 (0.42) FLT3USP30MAPK10MAPK8MAPK1
SCHEMBL12619136 0.80 MAPK10 (0.41) FLT3USP30MAPK10MAPK8
SCHEMBL13055060 0.79 MAP3K12 (0.41) MAPK10MAPK8
SCHEMBL801904 0.74 USP30 (0.43) FLT3USP30MAPK10MAPK8
SCHEMBL13055054 0.73 LCK (0.34)
SCHEMBL802069 0.73 MAPK10 (0.39) FLT3MAPK10MAPK8
SCHEMBL13055057 0.73 FADS1 (0.32) MAPK10MAPK8
SCHEMBL801907 0.71 FLT3 (0.45) FLT3MAPK10MAPK8
SCHEMBL13925111 0.71 AURKB (0.33)
SCHEMBL13055048 0.68 MAPK10 (0.34) MAPK10MAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7842712-B2 Indazolinone compositions useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-11-30 US disclosed
US-20090048250-A1 INDAZOLINONE COMPOSITIONS USEFUL AS KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED 2009-02-19 US disclosed
US-7262200-B2 Indazolinone compositions useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-08-28 US disclosed
US-7262200-B2 Indazolinone compositions useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-08-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090048250-A1 INDAZOLINONE COMPOSITIONS USEFUL AS KINASE INHIBITORS LCK, CDK2, MKNK2 FLT3 525/4885USP30 4040/4885MAPK10 435/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.