SCHEMBL13068993

SCHEMBL13068993

N=NC(=N)c1ccccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
KDM4E B2RXH2 6/20 0.48
LMNA P02545 5/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
NAPRT Q6XQN6 1/20 0.48
P4HTM Q9NXG6 1/20 0.48
ALDH1A1 P00352 3/20 0.47
KMT2A Q03164 4/20 0.44
GSK3B P49841 1/20 0.42
NPC1 O15118 5/20 0.40
RAB9A P51151 5/20 0.40
MAPT P10636 4/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
PKM P14618 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
GAA P10253 2/20 0.40
HPGD P15428 2/20 0.40
TP53 P04637 1/20 0.40
NFKB1 P19838 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26570939 0.84 CES2 (0.52) CES2CES1KDM4ELMNAL3MBTL1
SCHEMBL18087488 0.81 CES2 (0.48) CES2CES1KDM4ELMNAL3MBTL1
SCHEMBL3633578 0.81 CES2 (0.54) CES2CES1KDM4ELMNAL3MBTL1
SCHEMBL4144993 0.77
SCHEMBL11078493 0.77 CES2 (0.58) CES2CES1KDM4ELMNAL3MBTL1
SCHEMBL28782253 0.76 CES2 (0.48) CES2CES1KDM4ELMNAL3MBTL1
SCHEMBL23229581 0.75 CES2 (0.42) CES2CES1KDM4ELMNAL3MBTL1
SCHEMBL22606420 0.75 KDM4E (0.50) CES2CES1KDM4ELMNAL3MBTL1
SCHEMBL19413864 0.74 CES2 (0.45) CES2CES1KDM4ELMNAL3MBTL1
SCHEMBL1650571 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1485093-B1 DI-ARYL SUBSTITUTED TETRAZOLE MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR-5 MERCK SHARP & DOHME (US) 2010-11-03 EP disclosed