SCHEMBL13069643

SCHEMBL13069643

CN1CCCC2C[C@@H](NC(=O)c3n[nH]c4ccc(-c5cn(Cc6ccccc6)nn5)cc34)CC21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 19/20 0.60
DYRK1A Q13627 8/20 0.53
HIPK2 Q9H2X6 8/20 0.53
DAPK3 O43293 7/20 0.53
CDK5 Q00535 7/20 0.53
ROCK2 O75116 6/20 0.53
CLK2 P49760 6/20 0.53
PRKACA P17612 5/20 0.53
PAK4 O96013 5/20 0.53
PRKX P51817 5/20 0.53
MELK Q14680 5/20 0.53
MAP4K5 Q9Y4K4 5/20 0.53
PIM1 P11309 5/20 0.53
JAK2 O60674 4/20 0.53
MAPK13 O15264 4/20 0.53
CDK1 P06493 4/20 0.53
MAPK1 P28482 4/20 0.53
CSNK1D P48730 4/20 0.53
MAPK12 P53778 4/20 0.53
CSNK2A1 P68400 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13923963 0.87 CDC7 (0.63) CDC7DYRK1AHIPK2DAPK3CDK5
SCHEMBL3376687 0.86 CDC7 (0.65) CDC7DYRK1AHIPK2DAPK3CDK5
SCHEMBL3374092 0.86 CDC7 (0.65) CDC7DYRK1AHIPK2DAPK3CDK5
Formic Acid SCHEMBL2086823 0.84 CDC7 (0.62) CDC7DYRK1AHIPK2DAPK3CDK5
SCHEMBL2085428 0.80 CDC7 (0.56) CDC7DYRK1AHIPK2DAPK3CDK5
SCHEMBL2085431 0.80 CDC7 (0.56) CDC7DYRK1AHIPK2DAPK3CDK5
SCHEMBL13069184 0.79 DYRK1A (0.73) DYRK1AGSK3B
Formic Acid SCHEMBL2087409 0.78 CDC7 (0.53) CDC7DYRK1AHIPK2DAPK3CDK5
SCHEMBL13069595 0.77 GSK3B (0.58) DYRK1ACDK2GSK3B
SCHEMBL4289886 0.76 CDC7 (1.00) CDC7DYRK1AHIPK2DAPK3CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1742944-B1 INDOLES, 1H-INDAZOLES, 1,2-BENZISOXAZOLES, 1,2-BENZOISOTHIAZOLES, AND PREPARATION AND USES THEREOF MEMORY PHARM CORP (US) 2010-11-10 EP disclosed