SCHEMBL13069754

SCHEMBL13069754

C=C(Nc1cccc2c1C(=O)N(Cc1ccc(I)cc1)C2)c1ccc(Cl)s1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
F10 P00742 1/20 0.42
PARP1 P09874 1/20 0.39
HDAC1 Q13547 2/20 0.39
PREP P48147 4/20 0.37
ALDH1A1 P00352 1/20 0.36
NR1I2 O75469 1/20 0.35
UGCG Q16739 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8231433 0.92 F10 (0.48) F10PARP1HDAC1PREPALDH1A1
SCHEMBL3382279 0.90 F10 (0.49) F10PARP1HDAC1PREPALDH1A1
SCHEMBL8231182 0.86 F10 (0.43) F10PARP1HDAC1PREPALDH1A1
SCHEMBL8230002 0.86 F10 (0.41) F10PARP1HDAC1ALDH1A1NR1I2
SCHEMBL3382382 0.82 F10 (0.55) F10PARP1HDAC1PREPALDH1A1
SCHEMBL5781798 0.82 F10 (0.49) F10PARP1HDAC1PREPALDH1A1
SCHEMBL8231854 0.80 HDAC1 (0.39) F10HDAC1ALDH1A1HDAC7MAPK1
SCHEMBL8228040 0.78 F10 (0.45) F10PARP1PREPALDH1A1MAPK1
SCHEMBL3377544 0.78 F10 (0.51) F10PARP1HDAC1PREPALDH1A1
SCHEMBL5782990 0.77 F10 (0.55) F10PARP1HDAC1PREPALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2029586-B1 ISOINDOLIN-1-ONE-, ISOINDOLIN-3-ONE- AND ISOINDOLIN-1,3-DIONE-DERIVATIVES AND USE THEREOF BAYER SCHERING PHARMA AG (DE) 2010-11-24 EP disclosed