SCHEMBL13070871

SCHEMBL13070871

CCCCN(C)CCNC(=O)c1cccc(-c2nccc(OCCc3ccc(OC)c(OC)c3)n2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.47
TMEM97 Q5BJF2 2/20 0.47
SIGMAR1 Q99720 2/20 0.47
KDM5A P29375 1/20 0.45
MAPK1 P28482 2/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C8 P10632 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
CNR2 P34972 2/20 0.44
TP53 P04637 2/20 0.43
POLB P06746 2/20 0.43
MAPT P10636 3/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
THRB P10828 1/20 0.43
PKM P14618 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12919049 0.82 GPR52 (0.57) MAPK1CNR2TP53POLBMAPT
SCHEMBL12919079 0.81 GPR52 (0.56) OPRM1TMEM97SIGMAR1MAPK1TP53
SCHEMBL963885 0.81 F10 (0.51) SIGMAR1MAPK1TP53POLBMAPT
SCHEMBL12919083 0.80 GPR52 (0.56) TMEM97SIGMAR1MAPK1TP53POLB
SCHEMBL12919080 0.80 GPR52 (0.57) OPRM1TMEM97SIGMAR1MAPK1TP53
SCHEMBL958484 0.79 PTGDR (0.52) MAPK1POLBMAPTKDM4EALDH1A1
SCHEMBL959496 0.78 NPC1 (0.48) TP53MAPTKDM4EMEN1ALDH1A1
SCHEMBL12919098 0.78 GPR52 (0.58) OPRM1TMEM97SIGMAR1MAPK1TP53
SCHEMBL12919095 0.78 GPR52 (0.56) MAPK1TP53POLBMAPTKDM4E
SCHEMBL12919063 0.77 GPR52 (0.60) MAPK1TP53POLBMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2253618-A1 COMPOUND HAVING 6-MEMBERED AROMATIC RING Takeda Pharmaceutical Company Limited (JP) 2010-11-24 EP disclosed