SCHEMBL1307186

SCHEMBL1307186

CC(C)(C)OC(=O)N1CCC(NC/C(=C/c2ccc(C(=O)NO)cc2)COc2cccc3ccccc23)C1

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 2/20 0.70
USP30 Q70CQ3 6/20 0.40
HTR6 P50406 1/20 0.39
HDAC6 Q9UBN7 3/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC4 P56524 1/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
BRD4 O60885 1/20 0.39
SCN9A Q15858 1/20 0.38
CCR8 P51685 1/20 0.38
DGAT2 Q96PD7 2/20 0.37
PARP1 P09874 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1309133 0.92 P2RX3 (0.59) P2RX3USP30HTR6HDAC6HDAC4
SCHEMBL1308027 0.92 P2RX3 (0.61) P2RX3USP30HTR6KDM4EPKM
SCHEMBL1308028 0.92 P2RX3 (0.61) P2RX3USP30HTR6KDM4EPKM
SCHEMBL1308026 0.92 P2RX3 (0.61) P2RX3USP30HTR6KDM4EPKM
SCHEMBL2888069 0.89 P2RX3 (0.79) P2RX3HDAC6HDAC1HDAC4KDM4E
SCHEMBL2888065 0.89 P2RX3 (0.79) P2RX3HDAC6HDAC1HDAC4KDM4E
SCHEMBL2888072 0.89 P2RX3 (0.79) P2RX3HDAC6HDAC1HDAC4KDM4E
SCHEMBL1306813 0.87 P2RX3 (0.75) P2RX3USP30HTR6HDAC6HDAC4
SCHEMBL1306631 0.86 P2RX3 (0.71) P2RX3HDAC6HDAC1HDAC4KDM4E
SCHEMBL1306637 0.86 P2RX3 (0.71) P2RX3HDAC6HDAC1HDAC4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8053435-B2 Naphthalenyloxypropenyl derivatives having inhibitory activity against histone deacetylase and pharmaceutical composition comprising the same KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2011-11-08 US disclosed