SCHEMBL13076256

SCHEMBL13076256

C=C(Nc1nc(OC2CCNC2)ccc1N)C(=O)c1ccc(C#N)c(-c2c(C)nn(C)c2C)c1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.43
CCND1 P24385 1/20 0.43
CCND3 P30281 1/20 0.43
CDK6 Q00534 1/20 0.43
TBK1 Q9UHD2 3/20 0.34
JAK3 P52333 1/20 0.34
BCL9 O00512 5/20 0.32
CTNNB1 P35222 5/20 0.32
PAICS P22234 1/20 0.32
TOP2A P11388 3/20 0.31
HSP90AB1 P08238 1/20 0.31
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL112968 0.81 CDK4 (0.52) CDK4CCND1CCND3CDK6TBK1
SCHEMBL13075895 0.78 CDK4 (0.64) CDK4CCND1CCND3CDK6
SCHEMBL110672 0.71 CDK4 (0.55) CDK4CCND1CCND3CDK6TBK1
SCHEMBL111358 0.67 CDK4 (0.51) CDK4CCND1CCND3CDK6JAK1
SCHEMBL111791 0.67 CDK4 (0.48) CDK4CCND1CCND3CDK6
SCHEMBL13076282 0.66 CDK4 (0.43) CDK4CCND1CCND3CDK6JAK3
SCHEMBL111484 0.64 CDK4 (0.62) CDK4CCND1CCND3CDK6
SCHEMBL112413 0.61 CDK4 (0.53) CDK4CCND1CCND3CDK6
SCHEMBL111573 0.61 CDK4 (0.80) CDK4CCND1CCND3CDK6
SCHEMBL111458 0.61 CDK4 (0.58) CDK4CCND1CCND3CDK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125402-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS MODULATORS OF CYCLIN DEPENDENT KINASES NOVARTIS AG (CH) 2010-11-04 WO disclosed