SCHEMBL13077196

SCHEMBL13077196

Cc1cc(C)n(CC(=O)N2CCN(c3ccccc3-c3cccc(O)c3)CC2)n1

nearest known ligand 0.83

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 3/20 0.83
KCNH2 Q12809 1/20 0.83
ALDH1A1 P00352 4/20 0.47
LMNA P02545 3/20 0.44
TP53 P04637 2/20 0.42
KMT2A Q03164 1/20 0.42
POLB P06746 1/20 0.42
TSHR P16473 1/20 0.41
DPP4 P27487 1/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GAA P10253 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3732867 0.91 CXCR3 (0.88) CXCR3KCNH2ALDH1A1LMNATP53
SCHEMBL3735739 0.91 CXCR3 (0.88) CXCR3KCNH2ALDH1A1LMNATP53
SCHEMBL112559 0.91 CXCR3 (1.00) CXCR3KCNH2ALDH1A1LMNATP53
SCHEMBL3726536 0.89 CXCR3 (0.81) CXCR3KCNH2ALDH1A1LMNATP53
SCHEMBL3732650 0.89 CXCR3 (0.96) CXCR3KCNH2ALDH1A1LMNATP53
SCHEMBL3735286 0.88 CXCR3 (0.80) CXCR3KCNH2ALDH1A1LMNATP53
SCHEMBL3726827 0.87 CXCR3 (0.81) CXCR3KCNH2ALDH1A1LMNATP53
SCHEMBL3732576 0.87 CXCR3 (0.78) CXCR3KCNH2ALDH1A1LMNATP53
SCHEMBL3730735 0.87 CXCR3 (0.88) CXCR3KCNH2ALDH1A1LMNAKMT2A
SCHEMBL3739751 0.87 CXCR3 (0.77) CXCR3KCNH2ALDH1A1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010126811-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-04 WO disclosed