SCHEMBL13077288

SCHEMBL13077288

Cc1nc(NC[C@H](N)C(=O)OC(C)(C)C)c(C)c(N2CCC(c3ccc4c(n3)CCCC4)CC2)n1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.48
ITGB1 P05556 1/20 0.48
ITGAV P06756 1/20 0.48
ITGA5 P08648 1/20 0.48
ITGB5 P18084 1/20 0.48
ITGB6 P18564 1/20 0.48
ITGB8 P26012 1/20 0.48
TRPV3 Q8NET8 3/20 0.33
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
NR4A1 P22736 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5584350 0.88 ITGAV (0.62) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL277546 0.88 ITGAV (0.62) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL13039571 0.83 ITGB3 (0.47) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL13039567 0.81 ITGB3 (0.45) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL275146 0.81 ITGAV (0.57) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL276459 0.80 ITGAV (0.58) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL275460 0.79 ITGAV (0.52) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL5584347 0.77 ITGAV (0.69) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL12243894 0.77 ITGAV (0.65) ITGB3ITGB1ITGAVITGA5ITGB5
SCHEMBL275079 0.77 ITGAV (0.69) ITGB3ITGB1ITGAVITGA5ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825119-B2 Bone disorders such as osteoporosis, tumors and cardiovascular disorders; 4-(2-carboxy-2-Boc-aminoethylamino)-6-piperidinopyrimidines such as tert-butyl 2-benzyloxycarbonylamino-3-[2,5-dimethoxy-6-(4-[1,8]naphthyridin-2-yl-piperidin-1-yl)pyrimidin-4-ylamino]-propionate GALAPAGOS SAS (FR) 2010-11-02 US disclosed