SCHEMBL13077333

SCHEMBL13077333

CCc1c(NC[C@H](NCc2ccc(O)c(O)c2)C(=O)OC(C)(C)C)ncnc1N1CCC(c2ccc3c(n2)NCCC3)CC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 10/20 0.46
ITGB6 P18564 8/20 0.46
ITGB3 P05106 3/20 0.46
ITGB1 P05556 1/20 0.46
ITGA5 P08648 1/20 0.46
ITGB5 P18084 1/20 0.46
ITGB8 P26012 1/20 0.46
TRPV3 Q8NET8 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5584349 0.91 ITGAV (0.49) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL328003 0.91 ITGAV (0.47) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL328043 0.91 ITGB3 (0.44) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL5584194 0.90 ITGAV (0.46) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL14266376 0.89 ITGAV (0.44) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL328062 0.89 ITGAV (0.46) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL5584257 0.89 ITGAV (0.46) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL328139 0.88 ITGAV (0.44) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL328045 0.88 ITGAV (0.48) ITGAVITGB6ITGB3ITGB1ITGA5
SCHEMBL276367 0.88 ITGAV (0.48) ITGAVITGB6ITGB3ITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825119-B2 Bone disorders such as osteoporosis, tumors and cardiovascular disorders; 4-(2-carboxy-2-Boc-aminoethylamino)-6-piperidinopyrimidines such as tert-butyl 2-benzyloxycarbonylamino-3-[2,5-dimethoxy-6-(4-[1,8]naphthyridin-2-yl-piperidin-1-yl)pyrimidin-4-ylamino]-propionate GALAPAGOS SAS (FR) 2010-11-02 US disclosed