SCHEMBL13080682

SCHEMBL13080682

CC(C)C[C@@H](O)C(=O)N1CCN(c2nc(-c3ccccc3)nc3cc(C(=O)O)ccc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 2/20 0.46
GBA1 P04062 4/20 0.46
HDAC3 O15379 1/20 0.45
MTOR P42345 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
ABCG2 Q9UNQ0 4/20 0.45
KDM4E B2RXH2 1/20 0.44
STAT6 P42226 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TSHR P16473 1/20 0.44
LMNA P02545 2/20 0.43
ACHE P22303 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
ALOX15 P16050 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13080699 0.91 GBA1 (0.47) ACP1GBA1HDAC3MTORHDAC1
SCHEMBL13080784 0.91 GBA1 (0.47) ACP1GBA1HDAC3MTORHDAC1
SCHEMBL13080669 0.91 ACP1 (0.57) ACP1GBA1ABCG2KDM4ETSHR
SCHEMBL13080736 0.91 ACP1 (0.57) ACP1GBA1ABCG2KDM4ETSHR
SCHEMBL1623541 0.89 SMAD3 (0.52) GBA1HDAC3MTORHDAC1HDAC2
SCHEMBL1623546 0.89 SMAD3 (0.52) GBA1HDAC3MTORHDAC1HDAC2
SCHEMBL1624126 0.86 HDAC3 (0.40) HDAC3MTORHDAC1HDAC2HDAC6
SCHEMBL1624132 0.86 HDAC3 (0.40) HDAC3MTORHDAC1HDAC2HDAC6
SCHEMBL13080698 0.86 MEN1 (0.46) ACP1GBA1ABCG2KDM4ESTAT6
SCHEMBL13080697 0.83 CYP1A2 (0.49) ACP1GBA1ABCG2KDM4ESTAT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8283354-B2 Voltage gated sodium and calcium channel inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-10-09 US disclosed