SCHEMBL13080784

SCHEMBL13080784

Cc1ccc2c(N3CCN(C(=O)C(O)CC(C)C)CC3)nc(-c3ccccc3)nc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 5/20 0.47
ACP1 P24666 2/20 0.46
ABCG2 Q9UNQ0 3/20 0.44
MAPT P10636 1/20 0.44
KDM4E B2RXH2 1/20 0.44
STAT6 P42226 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
TSHR P16473 1/20 0.43
LMNA P02545 2/20 0.43
ACHE P22303 1/20 0.43
TP53 P04637 1/20 0.43
HDAC3 O15379 1/20 0.42
MTOR P42345 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
AKT1 P31749 1/20 0.41
NTSR1 P30989 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13080699 1.00 GBA1 (0.47) GBA1ACP1ABCG2MAPTKDM4E
SCHEMBL13080682 0.91 ACP1 (0.46) GBA1ACP1ABCG2MAPTKDM4E
SCHEMBL13080685 0.90 GBA1 (0.48) GBA1ACP1ABCG2MAPTKDM4E
SCHEMBL13080689 0.90 MAPT (0.47) GBA1ABCG2MAPTKDM4ESTAT6
SCHEMBL13080736 0.90 ACP1 (0.57) GBA1ACP1ABCG2MAPTKDM4E
SCHEMBL13080669 0.90 ACP1 (0.57) GBA1ACP1ABCG2MAPTKDM4E
SCHEMBL13080706 0.89 CYP1A2 (0.48) GBA1MAPTTSHRMEN1KMT2A
SCHEMBL13080708 0.89 GBA1 (0.47) GBA1ACP1ABCG2MAPTKDM4E
SCHEMBL13080688 0.89 GBA1 (0.47) GBA1ACP1ABCG2MAPTKDM4E
SCHEMBL1621278 0.88 MEN1 (0.49) GBA1MAPTKDM4ENPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8283354-B2 Voltage gated sodium and calcium channel inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-10-09 US disclosed