SCHEMBL13080752

SCHEMBL13080752

CCC(O)(CC)C(=O)NC1CCN(c2nc(-c3ccccc3)nc3ccccc23)CC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.58
TP53 P04637 5/20 0.53
MAPT P10636 4/20 0.53
KDM4E B2RXH2 1/20 0.53
ACP1 P24666 2/20 0.51
LMNA P02545 3/20 0.51
MEN1 O00255 1/20 0.51
USP2 O75604 1/20 0.51
HTT P42858 1/20 0.51
KMT2A Q03164 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
ABCG2 Q9UNQ0 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.47
ACHE P22303 1/20 0.47
GBA1 P04062 2/20 0.47
HSD17B10 Q99714 2/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
ALOX15 P16050 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13080756 0.91 TSHR (0.57) TSHRTP53MAPTKDM4EACP1
SCHEMBL13080744 0.91 TSHR (0.48) TSHRTP53MAPTKDM4EACP1
SCHEMBL13080745 0.89 TSHR (0.61) TSHRTP53MAPTKDM4EACP1
SCHEMBL1621972 0.89 SMAD3 (0.56) TSHRTP53MAPTKDM4ELMNA
SCHEMBL13080749 0.85 TSHR (0.57) TSHRTP53MAPTKDM4EACP1
SCHEMBL13080770 0.82 TSHR (0.47) TSHRTP53MAPTKDM4EACP1
SCHEMBL13080748 0.82 TSHR (0.58) TSHRTP53MAPTKDM4EACP1
SCHEMBL13080754 0.80 TSHR (0.56) TSHRTP53MAPTKDM4EACP1
SCHEMBL13080676 0.80 ABCG2 (0.57) TSHRMAPTKDM4EACP1LMNA
SCHEMBL1624722 0.80 SMAD3 (0.55) TSHRTP53MAPTKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8283354-B2 Voltage gated sodium and calcium channel inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-10-09 US disclosed