SCHEMBL13080920

SCHEMBL13080920

CCN(CCC(C)N1CCCCC1)C(=O)C(Cn1ccc(OCc2ccccc2)cc1=O)N(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 15/20 0.40
KCNH2 Q12809 6/20 0.39
MAPK14 Q16539 1/20 0.38
GHSR Q92847 2/20 0.37
UBE2M P61081 1/20 0.36
DCUN1D1 Q96GG9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3587238 0.77 MAPK14 (0.49) MCHR1KCNH2MAPK14
SCHEMBL3602692 0.77 MCHR1 (0.42) MCHR1KCNH2MAPK14
SCHEMBL4601498 0.72 MCHR1 (0.39) MCHR1KCNH2MAPK14
SCHEMBL3587241 0.70 MAPK14 (0.47) MCHR1KCNH2MAPK14
SCHEMBL7641512 0.67 MAPK14 (0.62) MCHR1MAPK14
SCHEMBL1365787 0.64 MCHR1 (0.71) MCHR1KCNH2MAPK14
SCHEMBL4488171 0.64 HTR6 (0.50) MCHR1MAPK14
SCHEMBL4484736 0.62 MAPK14 (0.76) MCHR1KCNH2MAPK14
SCHEMBL4470408 0.62 MAPK14 (0.64) MCHR1KCNH2MAPK14
SCHEMBL1523159 0.62 MAPK14 (0.67) MCHR1KCNH2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7842808-B2 calcitonin gene-related peptide receptors antagonists such as 4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperidine-1-carboxylic acid[2-(1,4-dioxa-8-aza-spiro [4.5]dec-8-yl)-1-(1H-indol-5-ylmethyl)-2-oxo-ethyl]-amide, used for treating headaches, pain, hot flashes or respiratory system disorders BRISTOL-MYERS SQUIBB COMPANY (US) 2010-11-30 US disclosed