SCHEMBL13080979

SCHEMBL13080979

COc1ccc(CC(C)NC(=O)N2CCC(N3Cc4ccccc4NC3=O)CC2)cn1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 18/20 0.54
CYP3A4 P08684 9/20 0.54
CALCA P06881 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3591393 0.91 CALCA (0.57) CALCRLCYP3A4CALCA
SCHEMBL13081133 0.90 CALCA (0.54) CALCRLCYP3A4CALCA
SCHEMBL14503776 0.90 CALCA (0.50) CALCRLCYP3A4CALCA
SCHEMBL3604161 0.88 CALCRL (0.72) CALCRLCYP3A4
SCHEMBL14503778 0.87 CALCRL (0.57) CALCRLCYP3A4
SCHEMBL3597734 0.84 CALCA (0.55) CALCRLCYP3A4CALCA
SCHEMBL3595749 0.81 CALCA (0.58) CALCRLCYP3A4CALCA
SCHEMBL13283564 0.81 CALCRL (0.76) CALCRLCYP3A4CALCA
SCHEMBL3754411 0.80 CALCRL (0.71) CALCRLCYP3A4
SCHEMBL27626938 0.80 CHRM4 (0.52) CALCRLCYP3A4CALCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7842808-B2 calcitonin gene-related peptide receptors antagonists such as 4-(2-Oxo-2,3-dihydro-benzoimidazol-1-yl)-piperidine-1-carboxylic acid[2-(1,4-dioxa-8-aza-spiro [4.5]dec-8-yl)-1-(1H-indol-5-ylmethyl)-2-oxo-ethyl]-amide, used for treating headaches, pain, hot flashes or respiratory system disorders BRISTOL-MYERS SQUIBB COMPANY (US) 2010-11-30 US disclosed
US-7754732-B2 Spirocyclic anti-migraine compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2010-07-13 US disclosed