SCHEMBL13086230

SCHEMBL13086230

O=C1Nc2ccc(I)cc2C(c2ccc(N3CC[C@@H](O)C3)nc2)=NC1Cc1ccccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 5/20 0.39
MCHR1 Q99705 1/20 0.35
MAPK8 P45983 2/20 0.35
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.35
ALB P02768 1/20 0.35
KMT2A Q03164 1/20 0.35
PGR P06401 1/20 0.34
MELK Q14680 1/20 0.34
IDH1 O75874 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2118497 0.92 CCKBR (0.47) CCKBRMCHR1MAPK8LMNAMEN1
SCHEMBL2118500 0.92 CCKBR (0.47) CCKBRMCHR1MAPK8LMNAMEN1
SCHEMBL2120515 0.88 CCKBR (0.50) CCKBRLMNAMEN1ALBKMT2A
SCHEMBL2117635 0.82 CCKBR (0.47) CCKBRMAPK8LMNAMEN1ALB
SCHEMBL2117626 0.81 CCKBR (0.51) CCKBRLMNAMEN1ALBKMT2A
SCHEMBL2119687 0.80 CCKBR (0.49) CCKBRLMNAMEN1ALBKMT2A
SCHEMBL2118545 0.79 CCKBR (0.49) CCKBRLMNAMEN1ALBKMT2A
SCHEMBL2119913 0.79 CNR2 (0.50) CCKBR
SCHEMBL13060992 0.79 CCKBR (0.50) CCKBRLMNAMEN1ALBKMT2A
SCHEMBL13086547 0.79 CHRM1 (0.40) CCKBRMCHR1MAPK8LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010121164-A2 1,4-BENZODIAZEPINONE COMPOUNDS AND THEIR USE IN TREATING CANCER THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2010-10-21 WO disclosed