SCHEMBL13086264

SCHEMBL13086264

Cc1ccc(NC(=O)C(N)C(C)C)nc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 12/20 0.60
MAPT P10636 4/20 0.60
XIAP P98170 1/20 0.51
BIRC2 Q13490 1/20 0.51
KDM4E B2RXH2 3/20 0.49
ALDH1A1 P00352 5/20 0.48
HPGD P15428 1/20 0.48
ATM Q13315 1/20 0.48
NPC1 O15118 11/20 0.48
SMN1; SMN2 Q16637 5/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
GAA P10253 2/20 0.47
TP53 P04637 2/20 0.47
GLA P06280 1/20 0.47
HSD17B10 Q99714 1/20 0.47
PKM P14618 1/20 0.47
HTT P42858 1/20 0.46
KEAP1 Q14145 1/20 0.45
NFE2L2 Q16236 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15986869 0.87 XIAP (0.64) RAB9AMAPTXIAPBIRC2KDM4E
SCHEMBL839860 0.85 RAB9A (0.66) RAB9AMAPTXIAPBIRC2KDM4E
SCHEMBL9891790 0.83 RAB9A (0.68) RAB9AMAPTXIAPBIRC2KDM4E
SCHEMBL839347 0.83 RAB9A (0.62) RAB9AMAPTXIAPBIRC2KDM4E
SCHEMBL839227 0.83 RAB9A (0.62) RAB9AMAPTXIAPBIRC2KDM4E
SCHEMBL839228 0.83 RAB9A (0.62) RAB9AMAPTXIAPBIRC2KDM4E
SCHEMBL21401471 0.81 RAB9A (0.64) RAB9AMAPTXIAPBIRC2KDM4E
SCHEMBL17409810 0.78 RAB9A (0.60) RAB9AMAPTXIAPBIRC2KDM4E
SCHEMBL5034164 0.76 RAB9A (0.72) RAB9AMAPTKDM4EALDH1A1NPC1
SCHEMBL7876929 0.76 POLB (0.63) RAB9AALDH1A1NPC1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010121164-A2 1,4-BENZODIAZEPINONE COMPOUNDS AND THEIR USE IN TREATING CANCER THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2010-10-21 WO disclosed