SCHEMBL13089176

SCHEMBL13089176

N[C@]12CN(CCCSc3nnc(-c4ccccc4)s3)C[C@@]1(c1ccc(C(F)(F)F)cc1)C2

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 15/20 0.45
KCNH2 Q12809 14/20 0.45
DRD2 P14416 12/20 0.45
GRIN2B Q13224 2/20 0.38
GRIN2A Q12879 1/20 0.38
HRH3 Q9Y5N1 1/20 0.35
CYP1A2 P05177 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2818179 0.81 DRD3 (0.68) DRD3KCNH2DRD2CYP1A2
Hydrochloric Acid SCHEMBL2845359 0.81 DRD3 (0.67) DRD3KCNH2DRD2CYP1A2
SCHEMBL13606600 0.70 DRD3 (0.58) DRD3KCNH2DRD2CYP1A2
SCHEMBL2818562 0.67 DRD3 (0.54) DRD3KCNH2DRD2CYP1A2
SCHEMBL2818705 0.67 DRD3 (0.64) DRD3KCNH2DRD2CYP1A2
SCHEMBL29864627 0.66 PTGS2 (0.48) GRIN2BGRIN2ACYP1A2ALDH1A1
Hydrochloric Acid SCHEMBL2844555 0.66 DRD3 (0.63) DRD3KCNH2DRD2CYP1A2
SCHEMBL2819960 0.66 DRD3 (0.67) DRD3KCNH2DRD2CYP1A2
SCHEMBL2821345 0.62 DRD3 (0.59) DRD3KCNH2DRD2CYP1A2
SCHEMBL2819404 0.62 DRD3 (0.59) DRD3KCNH2DRD2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891057-B1 AZABICYCLO[3.1.0]HEXANE DERIVAIVES AS DOPAMIN D3 RECEPTOR MODULATORS GLAXO GROUP LTD (GB) 2010-10-27 EP disclosed