SCHEMBL13093035

SCHEMBL13093035

CNNc1cc(C)nc2c(OCc3c(C)ccnc3Cn3cccc(C(F)(F)F)c3=O)cccc12

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 8/20 0.71
CYP3A4 P08684 4/20 0.70
CYP2C19 P33261 2/20 0.68
RORC P51449 11/20 0.42
CD38 P28907 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12711997 0.93 BDKRB2 (0.63) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL13448521 0.88 BDKRB2 (0.57) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL12712317 0.86 BDKRB2 (0.68) BDKRB2CYP3A4CYP2C19RORCCD38
SCHEMBL13146157 0.85 BDKRB2 (0.74) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL12711953 0.85 BDKRB2 (0.71) BDKRB2CYP3A4CYP2C19RORCCD38
SCHEMBL12711973 0.84 BDKRB2 (0.82) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL1563916 0.84 BDKRB2 (0.80) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL13146203 0.84 BDKRB2 (0.73) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL13145949 0.83 BDKRB2 (0.79) BDKRB2CYP3A4CYP2C19RORC
SCHEMBL12712293 0.83 BDKRB2 (0.77) BDKRB2CYP3A4CYP2C19RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2144897-B1 8-OXY-QUINOLINE DERIVATIVES AS BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-10-20 EP disclosed
WO-2008116620-A1 8-OXY-QUINOLINE DERIVATIVES AS BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2008-10-02 WO disclosed