SCHEMBL13093238

SCHEMBL13093238

C=C/C(Cl)=C(\NC)c1cc(C)nc2c(OCc3c(CNC(=O)C(C)C)ncc(F)c3C)cccc12

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 15/20 0.47
CYP3A4 P08684 2/20 0.47
ADORA2A P29274 3/20 0.35
CYP2C19 P33261 1/20 0.35
RORC P51449 1/20 0.34
CD38 P28907 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13093039 0.85 BDKRB2 (0.47) BDKRB2CYP3A4ADORA2ACYP2C19
SCHEMBL13145991 0.77 BDKRB2 (0.53) BDKRB2CYP3A4
SCHEMBL12711885 0.77 BDKRB2 (0.55) BDKRB2
SCHEMBL13145973 0.76 BDKRB2 (0.78) BDKRB2CYP3A4CYP2C19
SCHEMBL12712392 0.73 BDKRB2 (0.64) BDKRB2CYP3A4
SCHEMBL12711423 0.73 BDKRB2 (0.60) BDKRB2CYP3A4ADORA2ACYP2C19
SCHEMBL13093251 0.72 BDKRB2 (0.41) BDKRB2CYP3A4RORC
SCHEMBL12711400 0.72 BDKRB2 (0.52) BDKRB2CYP3A4CYP2C19
SCHEMBL13093092 0.72 BDKRB2 (0.61) BDKRB2CYP3A4ADORA2ACYP2C19CD38
SCHEMBL12711916 0.72 BDKRB2 (0.62) BDKRB2CYP3A4ADORA2ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2144897-B1 8-OXY-QUINOLINE DERIVATIVES AS BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-10-20 EP disclosed