SCHEMBL13093254

SCHEMBL13093254

Cc1cc(-c2[nH]ncc2C)c2cccc(OCc3c(Cl)cnc(O)c3Cn3cccc(N)c3=O)c2n1

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 20/20 0.62
CYP3A4 P08684 2/20 0.59
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13146266 0.90 BDKRB2 (0.59) BDKRB2CYP3A4CYP2C19
SCHEMBL1564610 0.90 BDKRB2 (0.73) BDKRB2CYP3A4CYP2C19
SCHEMBL14038571 0.85 BDKRB2 (0.51) BDKRB2
SCHEMBL12712322 0.85 BDKRB2 (0.51) BDKRB2
SCHEMBL1710376 0.82 BDKRB2 (0.74) BDKRB2CYP3A4CYP2C19
SCHEMBL1563908 0.78 BDKRB2 (0.62) BDKRB2CYP3A4CYP2C19
SCHEMBL13145116 0.78 BDKRB2 (1.00) BDKRB2
SCHEMBL12711441 0.77 BDKRB2 (0.88) BDKRB2CYP3A4CYP2C19
SCHEMBL1564611 0.76 BDKRB2 (0.59) BDKRB2CYP3A4
SCHEMBL1564948 0.75 BDKRB2 (0.48) BDKRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2144897-B1 8-OXY-QUINOLINE DERIVATIVES AS BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-10-20 EP disclosed
WO-2008116620-A1 8-OXY-QUINOLINE DERIVATIVES AS BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2008-10-02 WO disclosed