SCHEMBL13093267

SCHEMBL13093267

C#Cc1ccc(-c2cc(C)nc3c(OCc4c(Cl)cc(C)nc4Cn4ccc(=O)[nH]c4=O)cccc23)n1C

nearest known ligand 0.45

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 20/20 0.45
CYP3A4 P08684 2/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13146238 0.93 BDKRB2 (0.45) BDKRB2CYP3A4CYP2C19
SCHEMBL13093247 0.86 BDKRB2 (0.48) BDKRB2CYP3A4CYP2C19
SCHEMBL13093027 0.86 BDKRB2 (0.61) BDKRB2CYP3A4CYP2C19
SCHEMBL13146232 0.83 BDKRB2 (0.47) BDKRB2CYP3A4CYP2C19
SCHEMBL1563382 0.81 BDKRB2 (0.48) BDKRB2CYP3A4CYP2C19
SCHEMBL13146166 0.80 BDKRB2 (0.61) BDKRB2CYP3A4CYP2C19
SCHEMBL12711493 0.79 BDKRB2 (0.53) BDKRB2CYP3A4CYP2C19
SCHEMBL12711956 0.79 BDKRB2 (0.67) BDKRB2CYP3A4CYP2C19
SCHEMBL12711449 0.77 BDKRB2 (0.64) BDKRB2CYP3A4CYP2C19
SCHEMBL12711438 0.77 BDKRB2 (0.48) BDKRB2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2144897-B1 8-OXY-QUINOLINE DERIVATIVES AS BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-10-20 EP disclosed