Midodrine

Midodrine

SCHEMBL131436

COc1ccc(OC)c(C(O)CNC(=O)CN)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1D

The experimentally established mechanism targets of Midodrine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A known ✓ P35348 3/20 1.00
LMNA P02545 1/20 1.00
CYP1A2 P05177 1/20 1.00
TSHR P16473 1/20 1.00
CYP2C19 P33261 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
ADRA2A P08913 2/20 0.65
ADRB2 P07550 1/20 0.61
ADRB1 P08588 1/20 0.61
ADRB3 P13945 1/20 0.61
MTNR1A P48039 1/20 0.50
CYP2D6 P10635 2/20 0.49
MEN1 O00255 1/20 0.48
MAPK1 P28482 1/20 0.48
BLM P54132 1/20 0.48
KMT2A Q03164 1/20 0.48
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
ACHE P22303 1/20 0.45
SCN1A P35498 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(S)-Midodrine SCHEMBL6033144 1.00 ADRA1A (1.00) ADRA1ALMNACYP1A2TSHRCYP2C19
Midodrine SCHEMBL29367411 1.00 ADRA1A (1.00) ADRA1ALMNACYP1A2TSHRCYP2C19
(R)-Midodrine SCHEMBL30917926 1.00 ADRA1A (1.00) ADRA1ALMNACYP1A2TSHRCYP2C19
(R)-Midodrine SCHEMBL399213 1.00 ADRA1A (1.00) ADRA1ALMNACYP1A2TSHRCYP2C19
Midodrine SCHEMBL41463 0.99 ADRA1A (0.97) ADRA1ALMNACYP1A2TSHRCYP2C19
Midodrine SCHEMBL20899416 0.99 ADRA1A (0.97) ADRA1ALMNACYP1A2TSHRCYP2C19
Midodrine SCHEMBL20899425 0.99 ADRA1A (0.97) ADRA1ALMNACYP1A2TSHRCYP2C19
Midodrine SCHEMBL29368755 0.99 ADRA1A (0.97) ADRA1ALMNACYP1A2TSHRCYP2C19
Midodrine SCHEMBL41464 0.97 ADRA1A (0.95) ADRA1ALMNACYP1A2TSHRCYP2C19
Midodrine SCHEMBL20899432 0.96 ADRA1A (0.93) ADRA1ALMNACYP1A2TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 6566 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122094963-A Cardioprotective lipids and methods of use 2026-05-26 CN claimed
US-20260124148-A1 POLYPEPTIDE FORMULATIONS FOR ORAL DELIVERY BHAMIS RES LABORATORY PVT LTD (IN) 2026-05-07 US claimed
US-12617809-B2 Cardioprotective lipid and method of use SIGNPATH PHARMA, INC. (US) 2026-05-05 US claimed
US-20260027139-A1 TREATMENT OF SLEEP APNEA WITH A COMBINATION OF A CARBONIC ANHYDRASE INHIBITOR AND AN ALDOSTERONE ANTAGONIST VIVUS, INC. 2026-01-29 US claimed
US-12533321-B2 Polypeptide formulations for oral delivery Bhami's Research Laboratory, Pvt. Ltd. (IN) 2026-01-27 US claimed
US-20260000647-A1 Compositions, Formulations, And Methods Of Treating Neurodegenerative Diseases APPLIED COGNITION INC (US) 2026-01-01 US claimed
EP-4662311-A2 REVERSIR MOLECULES AND METHODS OF USE THEREOF Alnylam Pharmaceuticals, Inc. (US) 2025-12-17 EP claimed
US-12474326-B2 Treatment methods having reduced drug-related toxicity and methods of identifying the likelihood of patient harm from prescribed medications TABULA RASA HEALTHCARE, INC. (US) 2025-11-18 US claimed
US-12458610-B2 Pharmaceutical composition for treating or preventing diabetic cataract KOREA UNIVERSITY RESEARCH AND BUSINESS FOUNDATION (KR) 2025-11-04 US claimed
EP-4079311-B1 NMN AND DERIVATIVES FOR USE IN THE TREATMENT OF DEPRESSION AND/OR ANXIETY IN PATIENTS HAVING A FORM OF PARKINSONISM NUVAMID SA (CH) 2025-10-01 EP claimed
CN-1269811-A Polyanhydrides having therapeutically useful degradation properties RUTGERS THE STATE UNIV (US) 2000-10-11 CN claimed
EP-1032605-A1 POLYANHYDRIDES WITH THERAPEUTICALLY USEFUL DEGRADATION PRODUCTS Rutgers, The State University (US) 2000-09-06 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-6078834-A Device and method for detection and treatment of syncope PHARMATARGET, INC. (US) 2000-06-20 US claimed
WO-1999012990-A1 POLYANHYDRIDES WITH THERAPEUTICALLY USEFUL DEGRADATION PRODUCTS RUTGERS, THE STATE UNIVERSITY (US) 1999-03-18 WO claimed
US-5466466-A Therapeutic system for the retarded and controlled transdermal or transmucous administration of active substrates II LTS LOHMANN THERAPIE-SYSTEME GMBH & CO. KG (DE) 1995-11-14 US claimed
EP-0384266-B1 Therapeutic system for the sustained and controlled transdermal or transmucosal delivery of active agents LOHMANN THERAPIE SYST LTS (DE) 1994-07-20 EP claimed
US-5215751-A THERAPEUTIC SYSTEM FOR THE RETARDED AND CONTROLLED TRANSDERMAL OR TRANSMUCOUS ADMINISTRATION OF ACTIVE SUBSTANCES (I) LTS LOHMANN THERAPIE SYSTEME GMBH & CO. (DE) 1993-06-01 US claimed
EP-0384267-B1 THERAPEUTIC SYSTEM FOR THE SUSTAINED AND CONTROLLED TRANSDERMAL OR TRANSMUCOSAL DELIVERY OF ACTIVE AGENTS LTS Lohmann Therapie-Systeme GmbH & Co. KG (DE) 1993-05-26 EP claimed
EP-0164571-B1 SUSTAINED-RELEASE FORMS OF ALPHA-(2,5-DIMETHOXY PHENYL)-BETA-GLYCINAMIDOETHANOL AND PROCESS FOR THEIR PREPARATION CL PHARMA AKTIENGESELLSCHAFT (AT) 1990-06-27 EP claimed