SCHEMBL13145459

SCHEMBL13145459

COc1ccc(CN2CCc3nn(C)c4nc(N5CCN(c6ccccc6C)CC5)nc2c34)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.39
RECQL P46063 1/20 0.39
TSHR P16473 3/20 0.37
HTT P42858 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
KDM4E B2RXH2 2/20 0.37
LMNA P02545 2/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
GPR35 Q9HC97 2/20 0.37
ALOX15 P16050 2/20 0.37
ALDH1A1 P00352 3/20 0.37
ADRB2 P07550 1/20 0.37
GAA P10253 2/20 0.36
ATM Q13315 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HTR6 P50406 1/20 0.35
HRH4 Q9H3N8 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2815919 0.91 TSHR (0.43) TSHRHTTSMN1; SMN2KDM4ELMNA
SCHEMBL2812071 0.88 SMN1; SMN2 (0.43) TSHRHTTSMN1; SMN2KDM4ELMNA
SCHEMBL2809514 0.88 HTR6 (0.46) TSHRKDM4EHPGDHSD17B10ALOX15
SCHEMBL2811678 0.86 CCNE2 (0.39) TSHRHTTSMN1; SMN2KDM4ELMNA
SCHEMBL2810425 0.85 SMN1; SMN2 (0.44) NPC1TSHRHTTSMN1; SMN2KDM4E
SCHEMBL2809527 0.84 MAPT (0.45) NPC1SMN1; SMN2KDM4EHSD17B10ALDH1A1
SCHEMBL2810400 0.84 CFTR (0.46) NPC1TSHRHTTKDM4EHPGD
SCHEMBL2808261 0.81 TSHR (0.45) TSHRHTTSMN1; SMN2KDM4ELMNA
SCHEMBL2809446 0.81 TSHR (0.38) TSHRKDM4ELMNAHSD17B10ALDH1A1
SCHEMBL2814404 0.80 HRH4 (0.44) TSHRHTTSMN1; SMN2KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010114905-A1 PERI-FUSED PYRAZOLO-PYRIMIDINE COMPOUNDS ARQULE, INC. (US) 2010-10-07 WO disclosed