SCHEMBL13147657

SCHEMBL13147657

Nc1cc(-c2nccs2)nc(-c2nc(C(F)(F)F)cs2)n1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 4/20 0.41
HSP90AA1 P07900 1/20 0.41
SYK P43405 5/20 0.39
SRC P12931 4/20 0.39
ZAP70 P43403 4/20 0.39
CDK2 P24941 1/20 0.39
ADORA2A P29274 2/20 0.36
CYP1A1 P04798 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP1B1 Q16678 2/20 0.34
RAB9A P51151 1/20 0.34
CA2 P00918 1/20 0.33
CHKA P35790 1/20 0.33
CYP19A1 P11511 1/20 0.33
MAP4K4 O95819 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13147740 0.88 IDH1 (0.41) IDH1ADORA2ACA2CHKAADORA1
SCHEMBL578287 0.87 SYK (0.40) IDH1HSP90AA1SYKSRCZAP70
SCHEMBL1489975 0.82 HSP90AA1 (0.54) HSP90AA1SYKSRCZAP70CDK2
SCHEMBL14706466 0.81 IDH1 (0.37) IDH1HSP90AA1SYKSRCZAP70
SCHEMBL1926616 0.81 IDH1 (0.37) IDH1HSP90AA1SYKSRCZAP70
SCHEMBL13147656 0.81 KDM4E (0.47) CDK2ADORA2ACYP1A2RAB9ACYP19A1
SCHEMBL13147680 0.81 PTGS2 (0.40) IDH1HSP90AA1SYKSRCZAP70
SCHEMBL13147670 0.80 KDM4E (0.36) IDH1HSP90AA1CYP1A2
SCHEMBL13147662 0.80 IDH1 (0.36) IDH1HSP90AA1RAB9A
SCHEMBL13147742 0.80 IDH1 (0.37) IDH1ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118078-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed