SCHEMBL13147673

SCHEMBL13147673

N#Cc1csc(-c2cc(N)nc(-c3nc(C(F)(F)F)cs3)n2)c1

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 7/20 0.39
ATR Q13535 1/20 0.32
CA2 P00918 1/20 0.31
CHKA P35790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL578072 0.88 IDH1 (0.39) IDH1ATR
SCHEMBL13147740 0.82 IDH1 (0.41) IDH1CA2CHKA
SCHEMBL578236 0.81 IDH1 (0.36) IDH1
SCHEMBL13147659 0.79 IDH1 (0.35) IDH1
SCHEMBL13147660 0.78 IDH1 (0.39) IDH1CA2CHKA
SCHEMBL13147656 0.78 KDM4E (0.47)
SCHEMBL13147664 0.78 ALDH1A1 (0.44) IDH1CA2CHKA
SCHEMBL13147661 0.77 IDH1 (0.37) IDH1CA2CHKA
SCHEMBL13147742 0.77 IDH1 (0.37) IDH1
SCHEMBL1926969 0.76 PDE2A (0.37) IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118078-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed