SCHEMBL13148384

SCHEMBL13148384

C[N+](C)(Cc1ccc(NC(=O)c2cc3ccccc3s2)cc1)C1CCCCC1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 15/20 0.57
OPRM1 P35372 1/20 0.51
PTGDR2 Q9Y5Y4 1/20 0.47
F10 P00742 1/20 0.46
CCR5 P51681 1/20 0.46
CXCR5 P32302 1/20 0.45
CXCR3 P49682 1/20 0.45
TMIGD3 P0DMS9 1/20 0.44
ADORA2A P29274 1/20 0.44
ADORA1 P30542 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL5177249 0.99 CCR2 (0.56) CCR2OPRM1PTGDR2F10CCR5
Hydrochloric Acid SCHEMBL2906125 0.99 CCR2 (0.56) CCR2OPRM1PTGDR2F10CCR5
Hydrochloric Acid SCHEMBL313195 0.89 CCR2 (0.65) CCR2CCR5CXCR5CXCR3
Iodide SCHEMBL17555114 0.89 CCR2 (0.65) CCR2CCR5CXCR5CXCR3
SCHEMBL313427 0.78 NPC1 (0.58) CCR2
SCHEMBL13148385 0.78 MAPK1 (0.63) CCR2F10
Hydrochloric Acid SCHEMBL2906263 0.78 CCR2 (0.57) CCR2
Iodide SCHEMBL5178896 0.78 CCR2 (0.57) CCR2
Hydrochloric Acid SCHEMBL2907990 0.77 MAPK1 (0.62) CCR2F10
Iodide SCHEMBL17555183 0.77 MAPK1 (0.62) CCR2F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7799824-B2 Quaternary salt CCR2 antagonists ORAPHARMA, INC. (US) 2010-09-21 US disclosed