SCHEMBL13152145

SCHEMBL13152145

CCCn1c(-c2ccc(NS(=O)(=O)C3CC3)cc2)c(N)c2ccc(OC)cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SGK1 O00141 2/20 0.41
DYRK1A Q13627 2/20 0.39
BRPF1 P55201 2/20 0.39
PDE5A O76074 1/20 0.38
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
PRMT6 Q96LA8 2/20 0.36
ALDH2 P05091 1/20 0.36
PIK3CD O00329 1/20 0.36
MAP2K4 P45985 1/20 0.36
JAK1 P23458 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CNR2 P34972 1/20 0.35
PDE4A P27815 1/20 0.35
PRMT1 Q99873 1/20 0.34
PRMT8 Q9NR22 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13152587 0.94 DYRK1A (0.41) SGK1DYRK1ABRPF1PDE5AIDO1
SCHEMBL13151945 0.93 GRIK2 (0.40) SGK1BRPF1IDO1TDO2PRMT6
SCHEMBL13152186 0.92 KDM4E (0.43) SGK1DYRK1ABRPF1PDE5AIDO1
SCHEMBL13152481 0.90 SGK1 (0.41) SGK1BRPF1PDE5AIDO1TDO2
SCHEMBL13152254 0.89 SGK1 (0.39) SGK1BRPF1IDO1TDO2PRMT6
SCHEMBL13151731 0.88 CNR2 (0.42) SGK1BRPF1IDO1TDO2PRMT6
SCHEMBL13152062 0.87 DYRK1A (0.43) SGK1DYRK1ABRPF1PDE5AKDM4E
SCHEMBL13151897 0.87 DYRK1A (0.43) DYRK1APDE5AKDM4EALDH1A1MAPK1
SCHEMBL10097698 0.87 AR (0.41) SGK1DYRK1APDE5APRMT6
SCHEMBL10095986 0.86 DYRK1A (0.38) SGK1DYRK1ABRPF1PDE5AIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118009-A1 HCV INHIBITOR AND THERAPEUTIC AGENT COMBINATIONS PTC THERAPEUTICS, INC. (US) 2010-10-14 WO disclosed