SCHEMBL13152302

SCHEMBL13152302

Nc1ccc(-c2c(N)c3ccc(OC(F)F)cc3n2C2CCC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.36
PRKDC P78527 2/20 0.36
HTR3A P46098 1/20 0.33
GRM2 Q14416 1/20 0.33
MAT2A P31153 1/20 0.32
PDE7A Q13946 1/20 0.31
MTOR P42345 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
PRKACA P17612 1/20 0.30
RPS6KB1 P23443 1/20 0.30
GSK3B P49841 1/20 0.30
ROCK1 Q13464 1/20 0.30
DRD1 P21728 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10095958 0.86 CYP11B2 (0.41) PIK3CAPRKDCHTR3AGRM2MAT2A
SCHEMBL14466152 0.86 PRKACA (0.41) PIK3CAPRKDCHTR3APRKACARPS6KB1
SCHEMBL13152261 0.84 HRH3 (0.37) PIK3CAPRKDCNPC1RAB9AROCK1
SCHEMBL13152265 0.83 SGK1 (0.40) PIK3CAPRKDCHTR3AMTOR
SCHEMBL13152313 0.83 PIK3CA (0.36) PIK3CAPRKDCHTR3AMTORGSK3B
SCHEMBL10097497 0.82 DPP4 (0.37) PIK3CAPRKDCKMT2AGSK3B
SCHEMBL13152660 0.82 EPHX1 (0.43) NPC1RAB9AKMT2A
SCHEMBL13152247 0.82 NPC1 (0.39) PIK3CAPRKDCHTR3ANPC1RAB9A
SCHEMBL13153361 0.82 TDP1 (0.40) PIK3CAPRKDCMTORKMT2APRKACA
SCHEMBL13152697 0.81 SGK1 (0.40) PIK3CAPRKDCMTORGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118009-A1 HCV INHIBITOR AND THERAPEUTIC AGENT COMBINATIONS PTC THERAPEUTICS, INC. (US) 2010-10-14 WO disclosed