SCHEMBL13153251

SCHEMBL13153251

Fc1ccc(-n2c(CCc3cccc4cnccc34)nc3cc(F)ccc32)c(Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.62
AOC3 Q16853 1/20 0.37
PDE10A Q9Y233 1/20 0.36
P2RX7 Q99572 3/20 0.35
IDO1 P14902 1/20 0.34
CYP19A1 P11511 2/20 0.33
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
ACHE P22303 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
CYP17A1 P05093 1/20 0.33
CYP1A2 P05177 1/20 0.33
TRPV1 Q8NER1 1/20 0.32
TBXA2R P21731 1/20 0.32
DAO P14920 1/20 0.32
ROCK2 O75116 1/20 0.32
CCR2 P41597 1/20 0.32
ROCK1 Q13464 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3793533 0.83 GPBAR1 (0.88) GPBAR1AOC3P2RX7IDO1CYP17A1
SCHEMBL15426194 0.70 GPBAR1 (0.45) GPBAR1IDO1CYP19A1CYP11B1CYP11B2
SCHEMBL31258918 0.66 PDE10A (0.41) GPBAR1PDE10ACYP1A2
SCHEMBL3716494 0.62 GPBAR1 (0.57) GPBAR1CYP19A1CYP11B1CYP11B2
SCHEMBL11270913 0.61 CYP3A4 (0.55) PDE10ACYP1A2DAOROCK2CCR2
SCHEMBL6114531 0.61 KDM4E (0.50) PDE10ACYP1A2TRPV1DAOROCK2
SCHEMBL1830568 0.61 KDM4E (0.55) PDE10ACYP1A2TRPV1DAO
SCHEMBL27407502 0.61 CYP2D6 (0.50) PDE10ACYP1A2DAOROCK2ROCK1
SCHEMBL6965122 0.61 CYP3A4 (0.50) PDE10ACYP1A2TRPV1DAO
SCHEMBL3933037 0.60 CYP3A4 (0.53) PDE10ACYP1A2DAOROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010117090-A1 NOVEL ISOQUINOLINYLOXYMETHYL HETEROARYL DERIVATIVES BANYU PHARMACEUTICAL CO.,LTD. (JP) 2010-10-14 WO disclosed