SCHEMBL13178902

SCHEMBL13178902

O=C1C[C@H](NC(=O)[C@@H]2CCCN3C(=O)CCN(NC(=O)c4ccc(O)cc4)C(=O)N23)[C@H](OCc2ccccc2)O1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 11/20 0.48
CASP3 P42574 5/20 0.48
CASP8 Q14790 4/20 0.48
KLK7 P49862 1/20 0.39
MME P08473 1/20 0.35
ACE P12821 1/20 0.35
IL1B P01584 2/20 0.35
LCK P06239 2/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10200199 1.00 CASP1 (0.48) CASP1CASP3CASP8KLK7MME
SCHEMBL10247719 0.96 CASP1 (0.49) CASP1CASP3CASP8KLK7MME
SCHEMBL13139576 0.96 CASP1 (0.49) CASP1CASP3CASP8KLK7MME
SCHEMBL10199598 0.96 CASP1 (0.49) CASP1CASP3CASP8KLK7MME
SCHEMBL10200191 0.94 CASP1 (0.48) CASP1CASP3CASP8KLK7MME
SCHEMBL10263258 0.93 CASP1 (0.47) CASP1CASP3CASP8KLK7IL1B
SCHEMBL10200200 0.90 CASP1 (0.45) CASP1CASP3CASP8KLK7
SCHEMBL10200192 0.89 CASP1 (0.48) CASP1CASP3CASP8KLK7MME
SCHEMBL13139865 0.88 CASP1 (0.49) CASP1CASP3CASP8KLK7MME
SCHEMBL10200193 0.87 CASP1 (0.47) CASP1CASP3CASP8KLK7MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7790713-B2 Inhibitors of interleukin-1β converting enzyme VERTEX PHARMACEUTICALS INCORPORATED (US) 2010-09-07 US disclosed