SCHEMBL13190821

SCHEMBL13190821

Cn1nc2c(c1CC(=O)Nc1nc(-c3cc(Cl)ccc3F)cs1)c(=O)n(C)c(=O)n2C

nearest known ligand 0.71

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 20/20 0.71
TRPV4 Q9HBA0 7/20 0.54
TRPV3 Q8NET8 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL611387 0.89 TRPA1 (0.78) TRPA1TRPV4TRPV3
SCHEMBL612545 0.87 TRPA1 (0.71) TRPA1TRPV4TRPV3
SCHEMBL612052 0.87 TRPA1 (0.79) TRPA1TRPV4
SCHEMBL612021 0.86 TRPA1 (0.83) TRPA1TRPV4
SCHEMBL609319 0.84 TRPA1 (0.78) TRPA1TRPV4TRPV3
SCHEMBL612025 0.84 TRPA1 (0.75) TRPA1TRPV4TRPV3
SCHEMBL612471 0.83 TRPA1 (0.73) TRPA1TRPV4TRPV3
SCHEMBL1802273 0.83 TRPA1 (1.00) TRPA1TRPV4TRPV3
SCHEMBL480954 0.83 TRPA1 (0.88) TRPA1TRPV4
SCHEMBL611669 0.82 TRPA1 (0.76) TRPA1TRPV4TRPV3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010109287-A1 FUSED PYRIMIDINE-DIONE DERIVATIVES AS TRPA1 MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2010-09-30 WO disclosed