SCHEMBL13192017

SCHEMBL13192017

O=C1NC(=O)C2(Cc3ccc(I)cc3C2)N1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 2/20 0.42
CALCRL Q16602 6/20 0.41
TGM2 P21980 1/20 0.35
CES1 P23141 1/20 0.35
ADRA2A P08913 1/20 0.35
PNMT P11086 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
PDE7A Q13946 1/20 0.35
TSHR P16473 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CRBN Q96SW2 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
TNF P01375 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13055192 0.81 CALCRL (0.44) CALCRLADRA2APDE7APDE3BPDE3A
SCHEMBL16659357 0.81 TSHR (0.42) TDP2CALCRLADRA2APNMTADRA2B
SCHEMBL380001 0.80 CALCRL (0.41) TDP2CALCRLTSHRTDP1CRBN
SCHEMBL1727271 0.80 TDP2 (0.42) TDP2CALCRLADRA2APNMTADRA2B
SCHEMBL409009 0.78 TSHR (0.47) CALCRLPDE7ATSHRTDP1CRBN
SCHEMBL1726055 0.76 CALCRL (0.44) TDP2CALCRLPDE7ATDP1CRBN
SCHEMBL12698577 0.76 CALCRL (0.44) TDP2CALCRLPDE7ATDP1CRBN
SCHEMBL4629482 0.76 CALCRL (0.51) CALCRLCRBN
SCHEMBL12660698 0.75 CALCRL (0.45) TDP2CALCRLPDE7ACRBNPDE3A
SCHEMBL14614757 0.75 CALCRL (0.47) CALCRLCRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010107605-A1 CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2010-09-23 WO disclosed