SCHEMBL13192544

SCHEMBL13192544

C=C1NCCNC1Cc1cccc(F)c1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.40
PLG P00747 1/20 0.39
HTR2A P28223 1/20 0.38
SLC6A3 Q01959 2/20 0.38
SLC6A2 P23975 1/20 0.38
TRPA1 O75762 1/20 0.37
IDO1 P14902 2/20 0.36
AGXT P21549 2/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10153134 0.82 GLA (0.45) PLGHTR2ANPC1ALDH1A1SMN1; SMN2
SCHEMBL30406496 0.71 HTR2A (0.42) PLGHTR2ASLC6A3TRPA1ALDH1A1
SCHEMBL23115290 0.71 HTR2A (0.42) PLGHTR2ASLC6A3TRPA1ALDH1A1
SCHEMBL23115293 0.71 HTR2A (0.42) PLGHTR2ASLC6A3TRPA1ALDH1A1
SCHEMBL30406856 0.71 HTR2A (0.42) PLGHTR2ASLC6A3TRPA1ALDH1A1
SCHEMBL23222206 0.70 PLG (0.48) TAAR1PLGSLC6A3SLC6A2CHRM2
SCHEMBL13737199 0.68 SLC22A1 (0.41)
SCHEMBL10132275 0.68 POLB (0.58) PLGHTR2A
SCHEMBL20828166 0.68 POLB (0.58) PLGHTR2A
SCHEMBL3966432 0.67 GBA1 (0.62) PLGSLC6A3SLC6A2CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010107605-A1 CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2010-09-23 WO disclosed