SCHEMBL13198526

SCHEMBL13198526

CN1CCN(C(=O)[C@@H](COCc2ccccc2)NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 2/20 0.63
CTSS P25774 1/20 0.60
PPARG P37231 1/20 0.58
UGCG Q16739 13/20 0.58
CYP3A4 P08684 1/20 0.57
KLK7 P49862 2/20 0.53
KLK5 Q9Y337 2/20 0.53
KMT2A Q03164 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2538853 0.89 PPARA (0.60) PPARACTSSPPARGKLK7KLK5
SCHEMBL2538849 0.89 PPARA (0.60) PPARACTSSPPARGKLK7KLK5
SCHEMBL3746299 0.88 PPARA (0.62) PPARACTSSPPARGUGCGKLK7
SCHEMBL13291363 0.87 KMT2A (0.64) CTSSUGCGCYP3A4KMT2A
SCHEMBL27340724 0.87 KMT2A (0.64) CTSSUGCGCYP3A4KMT2A
SCHEMBL6582704 0.86 PPARA (0.59) PPARACTSSPPARGKLK7KLK5
SCHEMBL6582608 0.85 PPARA (0.60) PPARACTSSPPARGKLK7KLK5
SCHEMBL6582611 0.85 PPARA (0.60) PPARACTSSPPARGKLK7KLK5
SCHEMBL9090868 0.83 TACR1 (0.60) PPARACTSSPPARGUGCGCYP3A4
SCHEMBL9090873 0.83 TACR1 (0.60) PPARACTSSPPARGUGCGCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010091104-A1 GLUCOSYLCERAMIDE SYNTHASE INHIBITORS EXELIXIS, INC. (US) 2010-08-12 WO disclosed