SCHEMBL13208283

SCHEMBL13208283

Pc1ccc2c(n1)OCCNC2

nearest known ligand 0.43

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
APEX1 P27695 1/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2110694 0.79 APEX1 (0.32) APEX1HTR2AHTR2CHTR2BS1PR1
SCHEMBL10199960 0.79 HTR2A (0.37) APEX1HTR2AHTR2CHTR2BS1PR1
SCHEMBL10200081 0.79 CDK7 (0.37) APEX1HTR2AHTR2CHTR2BS1PR1
Hydrochloric Acid SCHEMBL2112542 0.78 HTR2A (0.36) APEX1HTR2AHTR2CHTR2BS1PR1
Hydrochloric Acid SCHEMBL2111829 0.78 CDK7 (0.36) APEX1HTR2AHTR2CHTR2BS1PR1
Hydrochloric Acid SCHEMBL2111995 0.78 APEX1 (0.31) APEX1HTR2AHTR2CHTR2B
SCHEMBL10200739 0.76 HTR2C (0.35) HTR2CHTR2BS1PR1
SCHEMBL2109252 0.76 S1PR1 (0.35) APEX1S1PR1
SCHEMBL10200689 0.76 NCF1 (0.32) S1PR1
SCHEMBL2110517 0.76 HTR2C (0.32) HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2213675-A1 PYRIDOOXAZEPINE DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2010-08-04 EP disclosed