SCHEMBL13220577

SCHEMBL13220577

O=C(NCCCNc1nsc2ccccc12)c1cccc(-c2ccccc2O)c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KISS1R Q969F8 4/20 0.42
SMYD2 Q9NRG4 1/20 0.42
HTR1A P08908 1/20 0.41
DRD2 P14416 1/20 0.41
HTR2A P28223 1/20 0.41
HTR7 P34969 1/20 0.41
HTR6 P50406 1/20 0.41
TP53 P04637 3/20 0.41
KCNA3 P22001 1/20 0.41
GPR52 Q9Y2T5 1/20 0.41
IKBKB O14920 1/20 0.40
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2979203 0.87 TP53 (0.45) KISS1RTP53MAPT
SCHEMBL2979166 0.84 FYN (0.43) KISS1RSMYD2TP53MAPT
SCHEMBL2976622 0.84 TP53 (0.47) SMYD2TP53KCNA3MAPT
SCHEMBL2976493 0.83 TP53 (0.44) KISS1RHTR1ADRD2HTR2AHTR7
SCHEMBL2972727 0.82 MAPT (0.47) TP53MAPT
SCHEMBL2966548 0.82 TP53BP1 (0.53) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL2969680 0.82 CDK4 (0.50) HTR1ADRD2HTR2AHTR7HTR6
SCHEMBL2977071 0.82 ALDH1A1 (0.53) TP53MAPT
SCHEMBL2971414 0.81 KCNH2 (0.49) TP53KCNA3MAPT
SCHEMBL2978922 0.81 LIMK1 (0.40) HTR1ADRD2HTR2AHTR7HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7776847-B2 Benzisothiazoles useful for treating or preventing HCV infection RIGEL PHARMACEUTICALS, INC. (US) 2010-08-17 US disclosed