SCHEMBL13220751

SCHEMBL13220751

COc1ccc(-c2ccc(C(=O)NCCCNc3nsc4c(I)cccc34)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
CDK4 P11802 1/20 0.46
CCND1 P24385 1/20 0.46
KMT2A Q03164 4/20 0.46
CFTR P13569 1/20 0.45
PTAFR P25105 1/20 0.43
HPGD P15428 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
ROCK2 O75116 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
PRKACA P17612 1/20 0.42
GSK3A P49840 1/20 0.42
GSK3B P49841 1/20 0.42
PRKX P51817 1/20 0.42
PRKCQ Q04759 1/20 0.42
ROCK1 Q13464 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2977401 0.89 KMT2A (0.48) NPC1RAB9ACDK4CCND1KMT2A
SCHEMBL2977008 0.89 NPC1 (0.47) NPC1RAB9ACDK4CCND1KMT2A
SCHEMBL2968665 0.85 NPC1 (0.44) NPC1RAB9ACDK4CCND1KMT2A
SCHEMBL2976173 0.83 USP30 (0.42) NPC1RAB9ACDK4CCND1KMT2A
SCHEMBL2961761 0.81 NPC1 (0.52) NPC1RAB9ACDK4CCND1KMT2A
SCHEMBL2977071 0.81 ALDH1A1 (0.53) RAB9AKMT2ACFTRPTAFRHPGD
SCHEMBL2972524 0.81 NPC1 (0.51) NPC1RAB9ACDK4CCND1KMT2A
SCHEMBL2979187 0.79 KMT2A (0.51) NPC1RAB9ACDK4CCND1KMT2A
SCHEMBL2977501 0.79 NPC1 (0.49) NPC1RAB9AKMT2ACFTRPTAFR
SCHEMBL2967147 0.79 KMT2A (0.57) NPC1RAB9AKMT2ACFTRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7776847-B2 Benzisothiazoles useful for treating or preventing HCV infection RIGEL PHARMACEUTICALS, INC. (US) 2010-08-17 US disclosed