SCHEMBL13233243

SCHEMBL13233243

CC(C)(C)OC(=O)NCCC(=O)Nc1cccc(O)c1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.60
CA2 P00918 2/20 0.60
SIRT5 Q9NXA8 1/20 0.52
NQO2 P16083 1/20 0.51
NLRP3 Q96P20 6/20 0.50
ALDH1A1 P00352 2/20 0.48
RAB9A P51151 2/20 0.48
NPC1 O15118 1/20 0.48
CYP1A2 P05177 2/20 0.47
MAPK1 P28482 2/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
MAPT P10636 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
SYK P43405 1/20 0.46
HDAC4 P56524 1/20 0.45
SUV39H2 Q9H5I1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14679432 0.87 CA1 (0.60) CA1CA2ALDH1A1RAB9ANPC1
SCHEMBL10845090 0.87 AURKB (0.53) CA1CA2SIRT5NQO2NLRP3
SCHEMBL4758303 0.86 CA1 (0.59) CA1CA2NQO2ALDH1A1CYP1A2
SCHEMBL16747675 0.86 GAA (0.61) CA1CA2ALDH1A1RAB9ANPC1
SCHEMBL15584781 0.86 CA1 (0.62) CA1CA2ALDH1A1NPC1CYP1A2
SCHEMBL4752807 0.86 CA1 (0.59) CA1CA2ALDH1A1CYP1A2MAPK1
SCHEMBL6274441 0.85 CA1 (0.58) CA1CA2ALDH1A1CYP1A2CYP3A4
SCHEMBL29459203 0.85 CA1 (0.58) CA1CA2ALDH1A1RAB9ANPC1
SCHEMBL10169791 0.85 CA1 (0.58) CA1CA2ALDH1A1RAB9ANPC1
SCHEMBL8692897 0.83 CA1 (0.66) CA1CA2SUV39H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198785-A1 OXIME DERIVATIVES USEFUL AS INHIBITORS OF HISTONE DEMETHYLASE KDM4C IEO - ISTITUTO EUROPEO DI ONCOLOGIA S.R.L. (IT) 2017-11-23 WO disclosed
US-7750151-B2 Inhibitors of Akt activity MERCK SHARP & DOHME CORP. (US) 2010-07-06 US disclosed
US-7750151-B2 Inhibitors of Akt activity MERCK SHARP & DOHME CORP. (US) 2010-07-06 US disclosed
US-20080280899-A1 Inhibitors of Akt Activity MERCK SHARP & DOHME CORP. 2008-11-13 US disclosed
US-20080280899-A1 Inhibitors of Akt Activity MERCK SHARP & DOHME CORP. 2008-11-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080280899-A1 Inhibitors of Akt Activity AKT1, AKT2, AKT3 CA1 1894/4885CA2 2592/4885SIRT5 1685/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.