SCHEMBL13243175

SCHEMBL13243175

CC(C)=C(C)c1c(C)ncnc1NC1CCN(C(C)c2cccc(F)c2)CC1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 6/20 0.38
CCL5 P13501 4/20 0.38
KCNH2 Q12809 1/20 0.37
P2RX3 P56373 1/20 0.37
ACKR3 P25106 4/20 0.37
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
MAP4K4 O95819 1/20 0.35
EGFR P00533 2/20 0.34
SOS1 Q07889 1/20 0.34
KDM4E B2RXH2 1/20 0.34
PAK1 Q13153 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1604053 0.77 MAPK1 (0.55)
SCHEMBL1604038 0.76 HTT (0.52) CNR1CNR2EGFR
SCHEMBL1604127 0.73 MEN1 (0.49) KDM4E
SCHEMBL1604243 0.72 MKNK1 (0.55) EGFR
Hydrochloric Acid SCHEMBL1920865 0.72 MEN1 (0.49) KDM4E
SCHEMBL1604186 0.67 MBTD1 (0.47) ACKR3
SCHEMBL12533526 0.64 GRIN2B (0.32) PAK1
SCHEMBL30341013 0.64 SLC6A2 (0.54) KCNH2
SCHEMBL19528703 0.63 MC4R (0.64) KCNH2
SCHEMBL1604737 0.62 MEN1 (0.50) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797099-B1 PIPERIDINYLAMINO-THIENO[2,3-D] PYRIMIDINE COMPOUNDS EPIX DELAWARE INC (US) 2010-08-11 EP disclosed